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Tirzepatide

The FDA and EMA approved Eli Lilly's Mounjaro (tirzepatide) peptide injection in May and July 2022, respectively. It is important to note that the identity of this peptide drug is a special GIP (glucose-dependent insulinotropic polypeptide) and GLP-1 (glucagon-like peptide-1) dual receptor agonist for the treatment of type II diabetes. Tirzepatide targets both GLP-1 and GIP receptors and is the first FDA-approved new drug. GLP-1/GIP dual receptor agonists, which exhibit better glycemic control and weight loss than selective GLP-1 receptor agonists. The amino acid sequence of tirzepatide is d on the endogenous GIP sequence, and the pharmacological effect on the GLP-1 receptor is comparable to that of endogenous GIP; The long half-life of tirzepatide of about 5 days can be achieved by dosing once a week. Tirzepatide was approved by the FDA on May 13, 2022 for the treatment of type 2 diabetes in adults, making it the first and only GIP and GLP-1 receptor agonist. Although tirzepatide is not currently available as a weight loss drug, it seems that it is only a matter of time from the current situation. Phase III Clinical SURMOUNT-1 (NCT04184622): Efficacy and Safety of tirzepatide Weekly in Participants With Obese or Overweight with Weight-Related Comorbidities: A Randomized, Double-Blind, Placebo-Controlled Trial Expected to be completed in the first half of 2024.